Part 5.  Radiopharmacy

1.   Mark the following statements True or False:

____   a) Tc-99m Sestamibi has a short biological half-life in the heart

____   b) Tc-99m Teboroxime has a short biological half-life in the heart

____   c) Tc-99m HMPAO has a long biological half-life in the brain

____   d) The tbiol of Tc-99m HSA in the blood pool is >Tc-99m RBC's

____   e) The tbiol of Tl-201 chloride in the body is less than 5 days

2. Match the renal agents listed below with their routes/percentages of excretion

______  Tc-99m DTPA                                   (A)    tubular secretion/glomerular filtration 50/50

______  Tc-99m MAG3                                   (B )   tubular secretion/glomerular filtration 80/20

______  I-131 Hippuran                                   (C)    glomerular filtration/tubular secretion 80/20

______ Tc-99m Glucoheptonate                    (D)    predominantly tubular binding

______ Tc-99m DMSA                                   (E)    tubular binding/glomerular filtration/tubular secretion 20/40/40

(F)    Tubular secretion 100%

(G)    Glomerular filtration 100%

 

3. Which of the following statements is incorrect?

a)   Tc-99m pertechnetate is distributed only in the blood pool

b)   Lesions detected on a cerebral radionuclide angiogram usually show increased uptake.

c)   Lesions detected on a delayed brain scan usually show decreased uptake.

d)   All of the above

e)   None of the above

 4. Which statement(s) is/are correct?

a)   Bone scanning is more sensitive than x-rays

b)   Bone scans detect metastatic disease prior to x-ray changes.

c)   Bone scans are less specific than x-rays

d)   a and b

e)   All of the above

5. The mechanism of radiopharmaceutical localization in lung scanning is:

a)   phagocytosis

b)   capillary blockade

c)   active transport

d)   adsorption to hydroxyapatite crystals

 6. Match the following:

a)   Ventilation lung scan                           _____ 1. Tc-99m macroaggregated albumin

b)   Perfusion lung scan                            _____ 2. Xenon-133

c)   Myocardial perfusion scan                  _____ 3. Thallium-201

d)   Myocardial infarct scan                       _____ 4. Tc-99m pyrophosphate

7. The mechanism of uptake of radiopharmaceutical in liver-spleen scanning is

a)   Particulate blockade

b)   Phagocytosis by the RE system

c)   Hydrolysis of the colloid particles by the hepatocytes

d)   b and c

e)   None of the above

 8.    The percent of Tc-99m sulfur colloid cleared from the circulation and the half-time of clearance are, respectively,

a)   50%, 8 min

b)   >90%, 2.5 min

c)   <10%, 3 min

d)   >90%, 8 min

e)   50%, 3 min

9. Clinical indications for spleen scanning with Tc-99m SC include

a) suspected lung abscess

b)   suspected splenic trauma and infarction

c)   evaluating the half-life of RBCs in splenic sequestration

d)   all of the above

e)   and c

10. Which of the following is/are suitable for thyroid imaging?

a)   Tc-99m sodium pertechnetate

b)   I-123 sodium iodide

c)   I-125 sodium iodide

d)   I-131 sodium iodide

11.    Pertechnetate and iodide uptake by the thyroid may be invalidated by which of the following?

a)    Angiographic contrast agents

b)    Propranolol

c)    Thyroid hormone ingestion

d)    a and c

e)    all of the above

12. Normal thyroid uptake of I-131 at 24 hours may be from

a)    3-10%

b)    7-30%

c)    >40%

d)    <2%

13. Which of the following radiopharmaceuticals is/are suitable for blood pool scanning?

      a)    Tc-99m sulfur colloid

b)    Tc-99m MAA

c)    Tc-99m tagged red blood cells

d)    Tc-99m tagged DTPA

e)    None of the above

 

14. Tl-201 is a useful cardiac imaging agent because of the following properties:

a)    It  is a potassium analog

b)    It localizes in acutely infarcted myocardium

c)    It is distributed proportional to relative blood flow.

d)    a and c only

e)    All of the above

15. The optimal time for detection of acute myocardial infarction by infarct avid agents is:

      a)    6 hours after onset of symptoms

b)    one week after onset of symptoms

c)    during chest pain

d)    24 to 72 hours after onset of symptoms

e)    during maximum exercise

16. Match the following

____1) Active transport                                   a)   Tc-99m MAA localizes in the lungs

____2) Capillary blockage                              b)   Fluorine-18 localizes in bone

____3) Phagocytosis                                      c)   In-111 Octreoscan

____4) Compartmental localization                d)   Iodine-131 localizes in thyroid

____5) Exchange diffusion                             e)   Tc-99m HSA localizes in blood pool

____6) Sequestration                                     f)    Tc-99m Sulfur Colloid localizes in RES cells

____7) Metabolic Trapping                             g)   In-111 Oncoscint

____8) Antigen/antibody reaction                   h)   Denatured Tc-99m RBC localizes in spleen

____9) Somatostatin receptor binding           I)     F-18 fluorodeoxyglucose

17.    The ideal diagnostic radiopharmaceutical has an effective half-life

a)   of 1 day

b)   1 to 1½ times the biological half‑life

c)   of 6 hours

d)   1 to 1½ times the length of time necessary to complete the test

18.    Which of the following is/are suitable for reducing pertechnetate prior to tagging to a chelating agent?        

 

b)   stannic ion (Sn4+)

c)   thallous ion (Tl1+) 

d)   mercuric ion (Hg2+) 

e)   none of the above

19. When can the effective half-life of a radioisotope equal the biological half‑life?

a)   when the physical half-life is very short

b)   when the physical half-life is infinitely long

c)   when the biological half-life is very short

d)   when the biological half-life is infinitely long

e)   when the biological and physical half-lives are equal

20.    We analyze all of  our Tc-99m radiopharmaceuticals for impurities. These include   

 

b)   free Tc, Mo99, Hydrolyzed Reduced Tc

c)   Al3+ , Mo99, Hydrolyzed Reduced Tc

d)   free Tc, Hydrolyzed Reduced Tc

e)   perchlorate, molybdate

21. Images of blood pool studies may be taken at what time post injection?

a)   minutes

b)   hours

c)   weeks

d)   a and b

e)   b and c

22.    Which of the following radiopharmaceuticals represents an example of compartmental localization?

a)   Tc - RBC

b)   Tc - HSA

c)   Tc - MAA

d)   a and b only

e)   all of the above

23.    Match radiation absorbed dose in right hand column with the item in the left hand column.

____ LD50 in humans (total body dose)                                              a)   O.l5R

____ LD100 in humans (total body dose)                                            b)   O.OlOR

____ Dose to thyroid gland of hyperthyroid patient                            c)   11,000R

following administration of 10 mCi of I‑131 NaI                         d)   500-550R

____ Whole body background if you live at sea level                         e)   1 x 106 R

____ Whole body background if you live in Denver                            f)    350R

____ Whole body dose from anterior chest film                                g)   0.3 R

 

24. Match particle size range with radiopharmaceutical

______ Tc-sulfur colloid                                                            a)   10-90 mm

______ Tc-MAA                                                                         b)   5-10 mm

______ Tc-MDP                                                                         c)   0.1-2 mm

______ Tc-MIAA                                                                         d)   no particles present

25.    Match number of particles of Tc-MAA to inject with patient population

______ Adult patient w/o pulmonary HTN                     a)    50,000

______ Adult patient w/ pulmonary HTN                       b)    350,000

______ 3 year old child                                                  c)    100,000

______ Neonate                                                             d)    150,000

26.    Three patients underwent dual Schillings Tests in which Co-57 labeled vitamin B12 bound to intrinsic factor and Co-58 vitamin B12 were administered. Match the results of the test with the proper diagnosis.

% excretion in 24 hrs.                                                           

Co-57 / Co-58                                                                                  Diagnosis:

 

____    21/18                                                                  a.  Malabsorption syndrome

____    4/3.6                                                                   b.  Normal

____    9/3                                                                      c.  Pernicious anemia

 

27     A patient underwent the first stage of a Schilling Test and the percent of administered Co-57 activity found in the urine at 24 hr post administration of the dose was 11.1%. The appropriate course of action is to

a.   Release the patient- test is complete

b.   Administer second stage of test

c.   Prescribe round of antibiotics, then repeat stage one

d.   Request an additional 24 hours of urine collection and pool specimens

28.    Match the procedure listed in column 1 with the typical adult dose in column 2

 

Column 1 (Procedure)                                                            Column 2 (Adult dose)           

 

_____ bone scan                                                                    a)    200 mCi

_____ perfusion lung scan                                                     b)    1 mCi

_____ thyroid uptake test                                                        c)    3 mCi

_____ liver scan                                                                      d)    5‑10 mCi

_____ thyroid therapy (Ca)                                                     e)    10‑15 mCi

_____ perfusion brain scan                                                    f)     15‑25 mCi

_____ tumor/abscess scan with Ga-67                                 g)    100‑150 mCi

_____ MUGA                                                                           h)    50 mCi

 

29. Answer True/False to the following statements regarding hepatobiliary agents

a)   Typical injected dose is 1 mCi

b)   In an emergency, one could substitute Tc‑99m Sulfur Colloid for Tc-DISIDA for use in hepatobiliary imaging

c)   If gallbladder accumulation of the DISIDA first appears on scan at 90 minutes post injection, this is a normal study.

d)   Gallbladder emptying is sometimes effected following admini­stration of a glass of milk.

e)   The -IDA ending on DISIDA stands for -imidodiacetic acid.

f)    Administration of IV morphine effectively empties the gall bladder

g)   typical administered dose of 3-8 mCi is based on body surface area

 

30. Match isotopes in left hand column with principal imaging energy (KeV) in right hand column

                Isotope                                                             Energy (KeV)

 

________  Tc-99m                                                                   a.  71

________  Co-57                                                                      b.  511

________  F-18                                                                        c.  122

________  I-131                                                                        d.  159

________ Tl-201                                                                      e.  140

________  I-123                                                                        f.  365

 

  31.  Match a radiopharmaceutical in the right hand column with the scan type in the left hand column.

______ Lung Perfusion                                                            A.    In-lll leukocytes

______ Meckels diverticulum                                                   B.    Tc-99m pertechnetate

______ Bone Marrow                                                               C.    I-123 mIBG

______ Parotid                                                                         D.    I-131 iodocholesterol

______ Abscess                                                                      E.    In-lll DTPA

______ Hepatobiliary                                                                F.    Tc-Disofenin

______ Glomerular Filtration                                                    G.    Tc-MAA

______ Tubular secretion                                                        H.    Tc-Glucoheptonate

______ Adrenal cortical tumor                                                 I.      Tc-DTPA

______ Thyroid uptake test                                                      J.     Tc-99m MAG3

______ Neuroblastoma                                                            K.    Ga-67 citrate

______ Insulinoma/glucagonoma                                            L.     Tc-99m RBC’s

______ Recurrent ovarian Ca                                                  M.    I-123 Sodium iodide

______ Hepatic hemangioma                                                  N.    Tc-99m sulfur colloid

O.    In-111 Octreoscan

P.    In-111 Oncoscint


 

32. What test animals were used for the original USP pyrogen test?

a. dogs

b. Limulus polyphemus

c. mice

d. rats

e. rabbits

33.      What advantage(s) does the Limulus Amebocyte Lysate test have over the “in vivo” pyrogen test?

a. very rapid

b. relatively inexpensive

c. very sensitive

d. all of the above

34.      Cold, non-radioactive vitamin B12 is given as part of the Schilling Test to:

a.   Initiate therapy in the patient

b.   Block B12 binding sites in the liver

c.   Reduce facial flushing

d.   Help differentiate between pernicious anemia and simple malabsorption

35.      The most common long-term adverse effect observed following the administration of an I-131 NaI therapy dose for treatment of Graves Disease is

a.   Adenocarcinoma of the thyroid

b.   Hypothyroidism

c.   Leukemia

d.   Pancytopenia

36.      The fraction of the pulmonary vasculature occluded by a typical dose of human albumin microspheres may be expected to be:

a.   0.1 or less

b.   0.01 or less

c.   0.001 or less

37.      The ideal particle size to use in man for lung scanning is:

a. 5-15 mm

b. 20-40 mm

c. 100-150 mm

d. 200-400 mm

38.      The chances of picking up functioning metastases from thyroid carcinoma by scan are increased by which of the following:

a. thyroidectomy

b. use of iodine‑123

c. use of pertechnetate

d. scanning at 72-96 hours

e. a and d

   39. The ideal radiopharmaceutical for clinical imaging studies has

         1.   an effective half‑life equal to 1½ times duration of test.

2.   an absence of particulate radiation

3.   a gamma energy of 100 to 250 keV

4.   a decay by isomeric transition

 

Answer:

a.   if only 1, 2 and 3 are correct

b.   if only 1 and 3 are correct

c.   if only 2 and 4 are correct

d.   if only 4 is correct

e.   if all are correct

40. The effective half-life of Tc-99m is

a.   6.02 hr

b.   12.04 hr

c.   6.02 hr x (½)10

d.   Not enough information to answer question

41. Within what % of the prescribed dose must the calibrated dose be?

a.   5%

b.   10%

c.   25%

d.   50%

42. The prescribed dose of Tl-201 chloride is 2.0 mCi. A technologist administers a 3.0 mCi dose since he has a very obese patient to inject. Whole body dose is estimated to be 3 R and no single organ receives more than 5 R. Which of the following describes the situation?

a.   Misadministration reportable only to the Nuclear Regulatory Commission